Open AccessChemistryMedicine
Fandi Sutanto, M. Konstantinidou, A. Dömling
2020.7.2RSC Medicinal Chemistry
tlooto Summary
In this review, a brief historic overview of covalent inhibitors is provided and recent advances focusing on developments in the last decade are summarized.
Abstract
In this review we provide a brief historic overview of covalent inhibitors and summarize recent advances focusing on developments in the last decade. Applications in challenging targets and future perspectives are also discussed.
Citation format
SUTANTO, Fandi; KONSTANTINIDOU, M.; DÖMLING, A. Covalent inhibitors: A rational approach to drug discovery. RSC Medicinal Chemistry, 2020, 11: 876–884.